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Table 2 Assessment of affinity for B-series bivalent inhibitors for proteins showing competition

From: Examining the influence of specificity ligands and ATP-competitive ligands on the overall effectiveness of bivalent kinase inhibitors

Gene Name Imatinib RB50 (μM) B-0 RB50 (μM) B-1 RB50 (μM) B-2 RB50 (μM)
ABL1 0.107 6.45 1.01 0.106
NQO2 4.93 6.71 >10 >10
  1. For affinity assessment of affinity for all kinases see Additional file 1