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Table 2 Assessment of affinity for B-series bivalent inhibitors for proteins showing competition

From: Examining the influence of specificity ligands and ATP-competitive ligands on the overall effectiveness of bivalent kinase inhibitors

Gene Name

Imatinib RB50 (μM)

B-0 RB50 (μM)

B-1 RB50 (μM)

B-2 RB50 (μM)

ABL1

0.107

6.45

1.01

0.106

NQO2

4.93

6.71

>10

>10

  1. For affinity assessment of affinity for all kinases see Additional file 1
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ISSN: 1477-5956