From: Examining the influence of specificity ligands and ATP-competitive ligands on the overall effectiveness of bivalent kinase inhibitors
Gene Name
Dasatinib RB50 (μM)
C-0 RB50 (μM)
C-1 RB50 (μM)
C-2 RB50 (μM)
ABL1
0.014
0.115
0.029
0.019
SRC
0.008
0.075
0.045
0.038
YES1
0.009
0.153
0.070
0.041
BTK
0.119
0.272
0.399
0.246
EPHB4
0.005
0.088
LYN
0.229
0.311